Structure and Function of GPCRs [E-Book] / edited by Guillaume Lebon.
Lebon, Guillaume, (editor)
1st edition 2019.
Cham : Springer, 2019
XIV, 289 pages 71 illustrations, 52 illustrations in color (online resource)
Topics in Medicinal Chemistry ; 30
Full Text
Table of Contents:
  • Structures of Non-rhodopsin GPCRs Elucidated Through X-Ray Crystallography
  • NMR Spectroscopy for the Characterization of GPCR Energy Landscapes
  • Structure and Activation Mechanism of GPCRs
  • Structure-Based Discovery of GPCR Ligands from Crystal Structures and Homology Models
  • Integration on Ligand and Structure Based Approaches in GPCRs
  • Biased Agonist Pharmacochaperones: Small Molecules in the Toolbox for Selectively Modulating GPCR Activity
  • Endosomal PTH Receptor Signaling Through cAMP and Its Consequence for Human Medicine
  • Structure and Function Studies of GPCRs by Site-Specific Incorporation of Unnatural Amino Acids
  • Fluorescent-Based Strategies to Investigate G Protein-Coupled Receptors: Evolution of the Techniques to a Better Understanding
  • Modulation of Metabotropic Glutamate Receptors by Orthosteric, Allosteric, and Light-Operated Ligands. .