JuLib | Articles & more - {"Medicinal chemistry."}

1

Poster

8,8'-Biflavone Analogues - Bioactivity Comparison of Dimers with Monomers

Klischan, Moritz
2023

2

Poster

Structural diversification of bioactive indole-based alkaloids using enzymatic methylation

Amariei, Diana-Alexandra
2023

3

Poster

Selective Biocatalytic Methylation of Dipeptides as a tool for Natural Product Synthesis

Haase, Mona
2023

4

Journal Article

7-[18F]Fluoro-8-azaisatoic Anhydrides: Versatile Prosthetic Groups for the Preparation of PET Tracers

Gröner, Benedikt
2023

Journal of medicinal chemistry, 66 (2023) 17, S. 12629−12644

OpenAccess OpenAccess

5

Journal Article

Innovative Non-PrP-Targeted Drug Strategy Designed to Enhance Prion Clearance

Colini Baldeschi, Arianna
2022

Journal of medicinal chemistry, 65 (2022) 13, S. 8998 - 9010

OpenAccess

6

Journal Article

Convenient PET-tracer production via SuFEx 18F-fluorination of nanomolar precursor amounts

Walter, Nils
2022

European Journal of Medicinal Chemistry European journal of medicinal chemistry, 237 237 (2022 2022) S. 114383 114383

Restricted Published on 2022-04-14. Available in OpenAccess from 2024-04-14.

7

Journal Article

Histamine H3 receptor antagonists with peptidomimetic (keto)piperazine structures to inhibit Aβ oligomerisation

Falkenstein, Markus
2021

Bioorganic & medicinal chemistry, 50 (2021) S. 116462 -

8

Journal Article

Discovery of new acetylcholinesterase inhibitors for Alzheimer’s disease: virtual screening and in vitro characterisation

David, Benoit
2021

Journal of enzyme inhibition and medicinal chemistry, 36 (2021) 1, S. 491 - 496

OpenAccess

9

Journal Article

All - d - Enantiomeric Peptide D3 Designed for Alzheimer’s Disease Treatment Dynamically Interacts with Membrane-Bound Amyloid-β Precursors

Bocharov, Eduard V.
2021

Journal of medicinal chemistry, 64 (2021) 22, S. 16464 - 16479

10

Journal Article

Radiosynthesis and Biological Evaluation of [18F]R91150, a Selective 5-HT2A Receptor Antagonist for PET-Imaging

Willmann, Michael
2021

ACS medicinal chemistry letters, 12 (2021) 5, S. 738 - 744

Published on 2021-04-01. Available in OpenAccess from 2022-04-01. Restricted

11

Journal Article

Design, synthesis and biological evaluation of Tozadenant analogues as adenosine A2A receptor ligands

Renk, Dana R.
2021

European Journal of Medicinal Chemistry European journal of medicinal chemistry, 214 214 (2021 2021) S. 113214 113214

Restricted Published on 2020-01-30. Available in OpenAccess from 2022-01-30.

12

Journal Article

Semisynthetic Analogs of the Antibiotic Fidaxomicin—Design, Synthesis, and Biological Evaluation

Dorst, Andrea
2020

ACS medicinal chemistry letters, 11 (2020) 12, S. 2414–2420

OpenAccess OpenAccess OpenAccess

13

Journal Article

Chiral Analogues of PFI-1 as BET Inhibitors and Their Functional Role in Myeloid Malignancies

Altenburg, Bianca
2020

ACS medicinal chemistry letters, 11 (2020) 10, S. 1928–1934

Published on 2020-04-02. Available in OpenAccess from 2021-04-02. Restricted Restricted

14

Journal Article

In silico/in vitro screening and hit evaluation identified new phenothiazine anti-prion derivatives

Zaccagnini, Ludovica
2020

European Journal of Medicinal Chemistry European journal of medicinal chemistry, 196 196 (2020 2020) S. 112295 112295

Published on 2020-04-08. Available in OpenAccess from 2022-04-08.

15

Journal Article

Converging a Knowledge-Based Scoring Function: DrugScore2018

Dittrich, Jonas
2019

Journal of chemical information and modeling, 59 (2019) 1, S. 509–521

Restricted Published on 2018-12-04. Available in OpenAccess from 2019-12-04. Restricted

16

Journal Article

Enantioselective total synthesis of altersolanol A and N

Mechsner, Bastian
2019

Bioorganic & medicinal chemistry, 27 (2019) 13, S. 2991 - 2997

17

Journal Article

Synthesis of peptoid-based class I selective histone deacetylase inhibitors with chemosensitizing properties

Krieger, Viktoria
2019

Journal of medicinal chemistry, 62 (2019) 24, S. 11260-11279

18

Journal Article

C-terminal Modulators of Heat Shock Protein of 90 kDa (HSP90): State of Development and Modes of Action

Bickel, David
2019

Bioorganic & medicinal chemistry, 27 (2019) 21, S. 115080

Published on 2019-08-26. Available in OpenAccess from 2021-08-26. Published on 2019-08-26. Available in OpenAccess from 2021-08-26.

19

Journal Article

Small-molecule inhibitors of nisin resistance protein NSR from the human pathogen Streptococcus agalactiae

Porta, Nicola
2019

Bioorganic & medicinal chemistry, 27 (2019) 20, S. 115079

Published on 2019-08-26. Available in OpenAccess from 2021-08-26. Published on 2019-08-26. Available in OpenAccess from 2021-08-26.

20

Journal Article

The tetrahydroxanthone-dimer phomoxanthone A is a strong inducer of apoptosis in cisplatin-resistant solid cancer cells

Wang, Chenyin
2019

Bioorganic & medicinal chemistry, 27 (2019) 19, S. 115044

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